Anastrozole is an indispensable aid to any athlete who uses anabolic steroids. Many anabolics can aromatize into the female sex hormone estradiol. Estradiol’s elevated levels cause a variety of unwanted effects, ranging from water retention and increased blood pressure to gynecomastia and poor libido. Anastrozole belongs to the group of aromatase inhibitors that can be used during a cycle of steroids in sports for the following purposes:
- Averting gynecomastia
- Increase in the level of testosterone in the blood
- Better muscle definition (by eliminating the negative effect of estrogens, which can lead to the formation of excess fat deposits)
- Prevention of hypertension
- Reduction of estrogenic suppression of the hypothalamus, pituitary gland, and testicles, which leads to a more rapid recovery of the body
Anastrozole for Men—Dosage and Using During Cycles
Using the drug should go hand in hand with a cycle of anabolic steroids. However, it’s unnecessary to hurry. First, athletes need to find out whether estradiol is high. They can do this by getting a blood test.
If there’s an increased concentration, athletes take Anastrozole tabs at a dosage of 0.25 to 0.5 mg every other day. In a week, again they have to do bloodwork. If the level of estradiol has returned to normal, athletes will continue to take the drug in the same dosage with the same frequency. However, if the level of the hormone is still high, the dosage and/or frequency should increase (0.25-0.5 mg every day).
After swallowing, the GI tract quickly absorbs the medication. Maximum plasma content is usually achieved within 60 minutes (in a fasted state). Food consumption somewhat hinders this impressive rate but does not influence the grade of absorption.
Anastrozole for Sale: Key Effects of the Drug
Anastrozole for men helps athletes to suppress the processes of aromatization in the body. In addition, the use of the medicament provides an increase in the level of endogenous T, provided there are no exogenous hormones in the body.
The effects of using Anastrozole in bodybuilding are:
- Removal of excess water, accumulated because of high estradiol, from the body
- Aromatization suppression, which lowers estradiol
- Increased levels of endogenous testosterone (if there are no external hormones in the body)
Anastrozole Side Effects: Undesirable Consequences of Taking Tabs
The following Anastrozole side effects occur often:
- Hot flashes
- Arthralgia (stiffness of the joints)
In addition, the drug may cause other unpleasant side effects, such as hair loss, allergic manifestations, nausea and vomiting, weariness, anorexia nervosa, hyperlipidemia, and bone discomfort.
Anastrozole 1 MG—Using for Medical Purposes
In postmenopausal women, estradiol (C18H24O2) is chiefly “manufactured” by transmuting androstenedione (4-androstenedione) to estrone through estrogen synthase CYP19A1 in peripheral tissues. Estrone (C18 steroid) is eventually turned into estradiol.
Reducing the level of circulating estradiol has beneficial effects for individuals suffering from breast cancer. Post menopause, the remedy at a daily dose of 1 mg suppressed estradiol by over 80% (as shown by highly sensitive tests). Therefore, the drug can be used for the following purposes:
Adjuvant therapy (given after the primary treatment) of stage 1 breast cancer with positive hormonal receptors in postmenopausal females
Neo-adjuvant therapy in locally advanced breast cancer (LABC)
Adjunct therapy of receptor-positive early invasive breast cancer
A 1 mg dosage is typically prescribed to treat the above diseases. Patients having mild-to-moderate end-stage renal disease (ESRD) do not require a dose adjustment. The same goes for people with mild liver diseases. Anastrozole is contraindicated for women during premenopause. Biochemical testing of the luteinizing hormone, follicle-stimulating hormone, and the level of estradiol should confirm the necessity.
The medicine is available in different countries under innumerable brands:
- Ai Da (Yangtze River Pharma)
- Altraz (Alkem)
- Amenur (GP Pharm)
- Anadex (medac)
- Anaprex (PHARMAGEN)
- Anaromat (Actavis)
- Egistrazol (Egis)
- Arilla (Mensana)
- Anastralan (PharmaSwiss)
- Anastrole RBX (Accord Healthcare Pty Ltd)
- Anastrozol by Cinfa, Cipla, Genericon, Genera, and Combix
- Aristu (Onko-Koçsel)
- Armistraz (Vitalchem)
- Azonet (Farmal)
- Enastros (Aurora)
- Griset (Genetic)
- Madelen (Rider)
- Xtrozol (Lambda)
- Zolkir (Pharmacenter)
Anastrozole for Bodybuilding—Buy Online and In Regular Drugstores
You can legally buy it online (or in a regular pharmacy) if you have a prescription from a licensed healthcare expert. It is a drug for females (when used in medicine). A version for males is available on the black market. Brands that are popularly used in athletics include Anatero (Lyka Labs), Armilon (Celon Laboratories), Femitraz (Lupin), Stazonex (Abbott), Qubol (Neon), and Xenosoul (Xeno).
Anastrozole—Price of the Medication
The medicament is available for sale at an affordable price—around $15.00 for a supply of 30 tablets. The underground cost of the drug can vary. For instance, 10 tabs of Qubol (1 mg) 10 is approximately 693 Indian Rupees (INR), about ten bucks. The cost of PMBC medication (from Miracalus Pharma) is 700 INR which is pretty much identical.