Anastrozole is an indispensable assistant to any bodybuilder who uses anabolic steroids. The vast majority of drugs have the ability to aromatize into the female sex hormone estradiol, the elevated level of which causes a variety of side effects, ranging from water retention & increased blood pressure to gynecomastia and lowering of libido. The drug belongs to the group of aromatase inhibitors that can be used during the cycle of steroids in sports with the following purposes:
1) prevention of gynecomastia;
2) increase in the level of anabolic hormones in the blood;
3) increase of the definition of the muscles (by eliminating the negative effect of estrogens, which can lead to the formation of excess fat deposits);
3) prevention of hypertension;
4) reduction of estrogenic suppression of the hypothalamus, pituitary gland, and testicles, which leads to a more rapid recovery of the body.
Anastrozole for men – dosage and using during cycles
The use of the drug should go in parallel with the cycle of anabolic steroids. However, it is not necessary to hurry. First, athletes need to find out if the level of estradiol is elevated. This can be done by performing blood tests.
If the concentration of estradiol in the blood is increased, athletes take Anastrozole tabs at a dosage of 0.25-0.5 mg every other day, or every two days. In a week again they have to take blood tests. If the level of estradiol returned to normal, athletes continue to take the drug in the same dosage with the same frequency. However, if the level of the hormone is still high, the athletes increase the dosage or start taking the drug more often (0.25-0.5 mg every day).
After ingestion, the medication is quickly absorbed from the gastrointestinal tract. The maximum concentration in the blood plasma is usually achieved within 2 hours (on an empty stomach). The food somewhat reduces the speed, but not the degree of absorption.
Anastrozole for sale – key effects of the drug
Anastrozole for men helps athletes to suppress the processes of aromatization in the body. In addition, the use of the medicament provides an increase in the level of its own testosterone, provided there is no exogenous hormones in the body.
The effects of using Anastrozole bodybuilding are as follows:
1) suppression of the aromatization process, therefore, a decrease in the level of estradiol;
2) the removal of excess water in the body, the retention of which is a consequence of the high level of estradiol.
3) increase the level of endogenous testosterone (if there are no external hormones in the body).
Anastrozole side effects – undesirable consequences of tabs taking
The following Anastrozole side effects occur quite often:
1) hot flashes;
3) arthralgia/stiffness of the joints;
8) skin rash;
In addition, the drug may cause some other side effects, such as hair loss, allergic reactions, nausea and vomiting, drowsiness, anorexia, hypercholesterolemia, bone pain, etc.
Anastrozole 1 mg – using for medical purposes
In postmenopausal women, estradiol is mainly produced by converting androstenedione to estrone through the aromatase enzyme complex in peripheral tissues. Estrone is subsequently transformed into estradiol. Reducing the level of circulating estradiol has beneficial effects for women with breast cancer. In postmenopausal women, a medication at a daily dose of 1 mg caused suppression of estradiol by more than 80% (as shown by highly sensitive tests). Therefore, the drug can be used for the following purposes:
- adjuvant therapy (given after the primary treatment) of early breast cancer with positive hormonal receptors in postmenopausal women;
- locally advanced breast cancer in postmenopausal women;
- adjuvant therapy of receptor-positive early invasive breast cancer in postmenopausal women.
For the treatment of the above diseases, 1 mg dosage should be used. Patients with mild to moderate renal dysfunction do not need a dose adjustment. Patients with mild violations of liver function do not need a dose adjustment either. Anastrozole should not be administered to women during premenopause. Menopause should be confirmed by biochemical testing (luteinizing hormone, follicle-stimulating hormone, and level of estradiol).
Anastrozole bodybuilding – buy online and in regular drugstores
You can buy online (or in regular pharmacy) this medicament legally if you have a prescription from a licensed healthcare expert. It is a drug for females (when using in medicine). A version for males is available on the black market.
Anastrozole – price of the medicament
The medicament is available for sale at an affordable price – around 15 dollars for a supply of 30 tablets. The cost of the drug at the black market can be lower.